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Abemaciclib methanesulfonate

CAT: 0931-T3111-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0931-T3111-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1231930-82-7
Target
CDK
Related Pathways
Cell Cycle/Checkpoint
Purity
0.9944
Bioactivity
Abemaciclib methanesulfonate (LY2835219) is a specific and effective inhibitor of CDK4 (IC50=2 nM) and CDK6 (IC50=10 nM) .
Smiles
CS(O)(=O)=O.CCN1CCN(Cc2ccc(Nc3ncc(F)c(n3)-c3cc(F)c4nc(C)n(C(C)C)c4c3)nc2)CC1
Molecular Formula
C27H32F2N8·CH4O3S
Molecular Weight
602.7
Shipping Conditions
Ice Packs
Storage Temperature
-20°C