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YM-430

CAT: 0931-T29183-01Size: 25 mgDry Ice: NoHazardous: No
CAT#:0931-T29183-01Size:25 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
153192-22-4
Target
Others|||Calcium Channel|||Adrenergic Receptor
Related Pathways
Others|||Metabolism|||GPCR/G Protein|||Membrane transporter/Ion channel|||Neuroscience
Bioactivity
YM-430 is a ?1 adrenergic receptor antagonist and a calcium channel antagonist. YM430 could be both an antianginal and antihypertensive agent. YM430 (10 (-8) -10 (-6) M) inhibited 3,4-diaminopyridine-induced rhythmic contractions with an IC50 value of 59.2 nM. In anesthetized rats, YM430 (10-100 mg/kg PO) inhibited arginine vasopressin-induced ST-segment depression with an IC50 value of 36.6 mg/kg PO.
Smiles
C(OCCCCNC[C@@H](COC1=CC=CC=C1)O)(=O)C=2[C@H](C(C(OC)=O)=C(C)NC2C)C3=CC(N(=O)=O)=CC=C3
Molecular Formula
C29H35N3O8
Molecular Weight
553.6
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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