YIL 781

• Target :

  GHSR

• Related Pathways :

  GPCR/G Protein

• Purity :

  0.993

• Bioactivity :

  YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 ?M) . YIL 781 improves glucose homeostasis in vivo and in vitro by blocking ghrelin secretion.

• Smiles :

  O=C1C=2C(N=C(C)N1C[C@@H]3CN(C(C)C)CCC3)=CC=C(OC4=CC=C(F)C=C4)C2

• Molecular Formula :

  C24H28FN3O2

• Molecular Weight :

  409.5

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  875258-85-8