YIL 781

• Target:

  GHSR

• Related Pathways:

  GPCR/G Protein

• Purity:

  0.993

• Bioactivity:

  YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 ?M) . YIL 781 improves glucose homeostasis in vivo and in vitro by blocking ghrelin secretion.

• Smiles:

  O=C1C=2C(N=C(C)N1C[C@@H]3CN(C(C)C)CCC3)=CC=C(OC4=CC=C(F)C=C4)C2

• Molecular Formula:

  C24H28FN3O2

• Molecular Weight:

  409.5

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  875258-85-8