Didesmethyl cariprazine

• Target:

  5-HT Receptor|||Dopamine Receptor

• Related Pathways:

  Neuroscience|||GPCR/G Protein

• Purity:

  0.997

• Bioactivity:

  Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors.

• Smiles:

  NC (=O) N[C@H]1CC[C@H] (CCN2CCN (CC2) c2cccc (Cl) c2Cl) CC1

• Molecular Formula:

  C19H28Cl2N4O

• Molecular Weight:

  399.36

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  839712-25-3