ARP-100

• Target :

  MMP

• Related Pathways :

  Proteases/Proteasome

• Purity :

  0.9834

• Bioactivity :

  ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM) . ARP-100 interacts with the S1' pocket of MMP-2 and exhibits anti-invasive properties in an in vitro invasion Matrigel model. ARP-100 has low inhibitory activity against MMP-1 (>50 ?M), MMP-3 (4.5 ?M), MMP-7 (>50 ?M) and MMP-9 (0.2 ?M) [1][2].

• Smiles :

  CC(C)ON(CC(=O)NO)S(=O)(=O)c1ccc(cc1)-c1ccccc1

• Molecular Formula :

  C17H20N2O5S

• Molecular Weight :

  364.42

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  704888-90-4