ZEN-3219

• Target:

  Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic

• Purity:

  0.9986

• Bioactivity:

  ZEN-3219 is a BET inhibitor, which has inhibitory effect on BRD4 (BD1), BRD4 (BD2) and BRD4 (BD1BD2) . ZEN-3219 has inhibitory effect on BRD4 (BD1), The IC50 values of BRD4 (BD2) and BRD4 (BD1BD2) were 0.48, 0.16 and 0.47 ?M, respectively. ZEN-3219 is a component of PROTAC molecule and can induce BRD4 degradation.

• Smiles:

  CC=1C(C2=CN(CC3=CC=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1

• Molecular Formula:

  C19H18N2O3

• Molecular Weight:

  322.36

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1952264-34-4