ZEN-3862

• Target:

  Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic

• Purity:

  0.971

• Bioactivity:

  ZEN-3862 (Willardiine) is an inhibitor of BET (IC50s of 0.16 and 0.13 ?M for BRD4 (BD1) and BRD4 (BD2), respectively) . ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.

• Smiles:

  CC=1C(C2=CN(CC3=CC(F)=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1

• Molecular Formula:

  C19H17FN2O3

• Molecular Weight:

  340.35

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1952264-33-3