Products for Research Use Only

GB-88

CAT: 0931-T11370Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T11370Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1416435-96-5
Target
Others, Protease-activated Receptor
Related Pathways
Others, GPCR/G Protein
Bioactivity
GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.
Smiles
CC[C@H](C)[C@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)c1ccno1)C(=O)N1CCC2(CC1)C=Cc1ccccc21
Molecular Formula
C32H42N4O4
Molecular Weight
546.7
Shipping Conditions
Ice Packs
Storage Temperature
-20°C