GB-88

• Target :

  Others|||Protease-activated Receptor

• Related Pathways :

  Others|||GPCR/G Protein

• Bioactivity :

  GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 ?M.

• Smiles :

  CC[C@H](C)[C@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)c1ccno1)C(=O)N1CCC2(CC1)C=Cc1ccccc21

• Molecular Formula :

  C32H42N4O4

• Molecular Weight :

  546.7

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1416435-96-5