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ERAP1-IN-1

CAT: 0931-T11221-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T11221-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
865273-97-8
Target
Others, Aminopeptidase
Related Pathways
Others, Metabolism
Purity
0.9895
Bioactivity
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor that allosterically activates ERAP1's hydrolysis of fluorogenic and chromogenic amino acid substrates, while competitively inhibiting its activity toward a nonamer peptide representative of physiological substrates.
Smiles
COc1ccc(cc1S(=O)(=O)Nc1cc(ccc1N1CCCCC1)C(F)(F)F)C(O)=O
Molecular Formula
C20H21F3N2O5S
Molecular Weight
458.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C