ERAP2-IN-1

CAT: 0931-MF-0042502-01Size: 50 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0042502-01Size:50 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2420551-38-6
Target
Others|||Aminopeptidase
Related Pathways
Others|||Metabolism
Bioactivity
ERAP2-IN-1 (compound 61) is a non-competitive inhibitor of ERAP2 that specifically inhibits its hydrolytic activity, with an IC50 of 27 ?M for Arg-AMC hydrolysis and an IC50 of 44 ?M for model peptide hydrolysis.
Smiles
N(S(=O)(=O)C1=C(OC)C=CC(C(O)=O)=C1)C2=C(C=C(C(F)(F)F)C=C2)N3CCCCC3
Molecular Formula
C20H21F3N2O5S
Molecular Weight
458.45
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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