PDK1/Akt/Flt Dual Pathway Inhibitor

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Cas number

331253-86-2
Chemical s molecular weight

224.18
Chemical s main applications

PDK1/Akt/Flt Dual Pathway Inhibitor is a cell-permeable compound that selectively induces apoptosis.
Chemical s formula

C10H4N6O
Physical properties

No Data Available
Melting temperature

No Data Available
Boiling temperature

No Data Available
Chemical s soluble in

No Data Available
Stability conditions

No Data Available
Storage

No Data Available
Chemical s specifications
Test

The duality of this product lies in it's dual specificity to the gene, pH or protein. Mainly in phosphorylation by specific phosphatases.
Description

Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.

Identity

HGNC:8809
Gene

PDK1
Long gene name

pyruvate dehydrogenase kinase 1
Synonyms gene name
- pyruvate dehydrogenase kinase, isoenzyme 1
- pyruvate dehydrogenase kinase, isozyme 1
GenBank acession
- L42450
Locus

2q31.1
Discovery year

1996-08-14
Entrez gene record

5163
Pubmed identfication
- 7499431
RefSeq identity
- NM_002610
VEGA ID

OTTHUMG00000132285