GSK852

CAT: 0804-HY-115867-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0804-HY-115867-01Size:1 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
GSK852 is a highly potent, second bromodomain (BD2) -selective, bromo and extra-terminal domain (BET) inhibitor (pIC50 = 7.9) .
CAS Number
[2305842-30-0]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gsk852.html
Purity
99.62
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
O=C(C1=CC(C(NC)=O)=C2OC[C@](C3=CC=CC=C3)(C)C2=C1)N[C@H]4[C@]5([H])C[C@@H](O)C[C@@]54[H]
Molecular Formula
C24H26N2O4
Molecular Weight
406.47
References & Citations
[1]Lucas SCC, et al. Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2) -Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors. J Med Chem. 2021 Aug 12;64 (15) :10711-10741.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-119608-01GSK854
HY-150760GSK5852
HY-145347GSK232
HY-100339-01GSK583
HY-111941-01GSK8612
HY-19540-01GSK864
HY-132880-01GSK251
HY-100220-01GSK6853
HY-153782GSK878
HY-107477-01GSK8573

Alternative Products

CatalogName
BA4742-5GSK852
A24410-1GSK852 1mg
A24410-10GSK852 10mg
A24410-50GSK852 50mg
A24410-5GSK852 5mg

Popular Products