17β-HSD1-IN-1

17β-HSD1-IN-1

• CAS Number: 2760791-96-4
• UNSPSC Description: 17β-HSD1-IN-1 (Compound 1) is a highly selective 17β-HSD1 inhibitor with IC50s of 5.6 and 3155 nM for 17β-HSD1 and 17β-HSD2, respectively. 17β-HSD1-IN-1 can be used for the research of non-small cell lung cancer (NSCLC)[1].
• Target Antigen: 17β-HSD
• Type: Reference compound
• Related Pathways: Metabolic Enzyme/Protease
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/17β-hsd1-in-1.html
• Solubility: DMSO : 100 mg/mL (ultrasonic)
• Smiles: CC1=CC=CC=C1N(C(C2=CC=C(O2)C3=CC(C)=C(C(C)=C3)O)=O)C
• Molecular Weight: 335.40
• References & Citations: [1]Emanuele M Gargano, et al. 17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer. ACS Med Chem Lett. 2021 Nov 18;12(12):1920-1924.
• Shipping Conditions: Room Temperature
• Clinical Information: No Development Reported