Products for Research Use Only

RL5a

CAT: 0804-HY-138886-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-138886-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
RL5a (compund C23) is a SETD8 inhibitor[1].
CAS Number
133671-66-6
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/rl5a.html
Purity
99.6
Solubility
DMSO : 40 mg/mL (ultrasonic; warming)
Smiles
CN(C)CCNC1=CC(C2=CC=CO2)=NC3=CC=CC=C13
Molecular Formula
C17H19N3O
Molecular Weight
281.35
References & Citations
[1]Gardner NJ, et al. The High-Affinity Interaction between ORC and DNA that Is Required for Replication Licensing Is Inhibited by 2-Arylquinolin-4-Amines. Cell Chem Biol. 2017 Aug 17;24 (8) :981-992.e4.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported