GGTI-2133
CAT:
804-HY-12369-04
Size:
50 mg
Price:
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
GGTI-2133
- CAS Number: 191102-79-1
- UNSPSC Description: GGTI-2133 is an inhibitor for geranylgeranyltransferase I (GGTase-I) with an IC50 of 38 nM. GGTI-2133 inhibits the geranylation of Rap-1A with an IC50 of 10 μM[1].
- Target Antigen: Others
- Type: Reference compound
- Related Pathways: Others
- Field of Research: Inflammation/Immunology
- Assay Protocol: https://www.medchemexpress.com/ggti-2133.html
- Purity: 98.38
- Solubility: DMSO : 100 mg/mL (ultrasonic)
- Smiles: CC(C)C[C@@H](C(O)=O)NC(C1=CC=C(NCC2=CN=CN2)C=C1C3=C4C=CC=CC4=CC=C3)=O
- Molecular Weight: 456.54
- References & Citations: [1]Vasudevan A, et al., Potent, highly selective, and non-thiol inhibitors of protein geranylgeranyltransferase-I. J Med Chem. 1999 Apr 22;42(8):1333-40.
- Shipping Conditions: Blue Ice
- Storage Conditions: -20°C, 3 years (Powder)
- Clinical Information: No Development Reported