CMPD-1

CAT: 0026-B2991-5Size: 5 mgDry Ice: NoHazardous: No
CAT#:0026-B2991-5Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
MK2a inhibitor is a substrate-selective inhibitor of p38α MAPK that selectively inhibits p38α-dependent phosphorylation of mitogen-activated protein kinase-activated protein kinase 2 (MK2a) with a K(i)(app) of 330 nM. It does not inhibit the phosphorylation of ATF-2 and MBP. It inhibits proliferation of U87, A172, and U251 glioblastoma cells with EC₅₀ values of 0.6-1 μM by inhibition of tubulin polymerization and induction of apoptosis.
Shipping Conditions
RT
Storage Conditions
-20ºC
Shelf Life
36 months