Brequinar Sodium
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


Brequinar Sodium
Description:
Brequinar sodium is a potent and selective dihydroorotate dehydrogenase (DHODH) inhibitor (IC50 = ~20 nM). Blocks de novo pyrimidine biosynthesis. Displays minimal inhibition against a panel of >400 kinases. Triggers differentiation of AML cell lines. Causes differentiation and depletion of leukemia-initiating cells in vivo. Antimetabolite.Shipping Conditions:
Gel PackStorage Conditions:
-20ºCShelf Life:
36 months
