Brequinar Sodium

CAT:
26-B2637-5
Size:
5 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
Brequinar Sodium - image 1

Brequinar Sodium

  • Description:

    Brequinar sodium is a potent and selective dihydroorotate dehydrogenase (DHODH) inhibitor (IC50 = ~20 nM). Blocks de novo pyrimidine biosynthesis. Displays minimal inhibition against a panel of >400 kinases. Triggers differentiation of AML cell lines. Causes differentiation and depletion of leukemia-initiating cells in vivo. Antimetabolite.
  • Shipping Conditions:

    Gel Pack
  • Storage Conditions:

    -20ºC
  • Shelf Life:

    36 months