PDE10A-IN-3

CAT:
804-HY-158237
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  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
PDE10A-IN-3 - image 1

PDE10A-IN-3

  • UNSPSC Description:

    PDE10A-IN-3 (Compound 8a) is an inhibitor of phosphodiesterase 10A (PDE10A). PDE10A-IN-3 can be used in schizophrenia research[1].
  • Target Antigen:

    Phosphodiesterase (PDE)
  • Type:

    Reference compound
  • Related Pathways:

    Metabolic Enzyme/Protease
  • Applications:

    Neuroscience-Neuromodulation
  • Field of Research:

    Neurological Disease
  • Assay Protocol:

    https://www.medchemexpress.com/pde10a-in-3.html
  • Solubility:

    10 mM in DMSO
  • Smiles:

    COC1=CC2=NC=NC(N3CC(C4=CC=CC=C4)CCC3)=C2C=C1OCCC5=NC6=CC=CC=C6C=C5
  • Molecular Weight:

    490.60
  • References & Citations:

    [1]Conrad J, et al. Model of P-Glycoprotein Ligand Binding and Validation with Efflux Substrate Matched Pairs. J Med Chem. 2024 Apr 11;67(7):5854-5865.
  • Shipping Conditions:

    Room temperature
  • Clinical Information:

    No Development Reported
  • CAS Number:

    1006889-85-5