BPR1J-097
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


BPR1J-097
UNSPSC Description:
BPR1J-097 is a novel potent FLT3 inhibitor with an IC50 of 11 nM.Target Antigen:
FLT3Type:
Reference compoundRelated Pathways:
Protein Tyrosine Kinase/RTKApplications:
Cancer-Kinase/proteaseField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/BPR1J-097.htmlSolubility:
10 mM in DMSOSmiles:
O=C(NC1=NNC(C2=CC=CC(NS(=O)(C3=CC=CC=C3)=O)=C2)=C1)C4=CC=C(N5CCN(C)CC5)C=C4Molecular Weight:
516.61References & Citations:
[1]Lin WH, et al. BPR1J-097, a novel FLT3 kinase inhibitor, exerts potent inhibitory activity against AML. Br J Cancer. 2012 Jan 31;106(3):475-81.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
1327167-19-0
