PKCζ-IN-1

CAT:

804-HY-120497-01

Size:

5 mg

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CAS Number: 1132609-87-0
UNSPSC Description: PKCζ-IN-1 is a compound that inhibits PKCζ and CDK2, showing an IC50 value of 5.18 nM for PKCζ and 1.04 μM for CDK2, with significant selectivity of 200-fold. PKCζ-IN-1 can reduce the activity of CDK2 while inhibiting PKCζ.
Target Antigen: CDK; PKC
Type: Reference compound
Related Pathways: Cell Cycle/DNA Damage;Epigenetics;TGF-beta/Smad
Field of Research: cancer
Assay Protocol: https://www.medchemexpress.com/pkcζ-in-1.html
Purity: 99.1
Smiles: CN(CC1)CCN1C2=CC=CC3=C2NC(C4=NNC5=C4C=CC(C6=CC=C(N)C=C6)=C5)=N3
Molecular Weight: 423.51
References & Citations: [1]2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: Design and synthesis of a potent and isoform selective PKC-f inhibitor
Shipping Conditions: Blue Ice
Storage Conditions: -20°C, 3 years (Powder)
Clinical Information: Launched

Cat	Name
HY-120497-02	PKCζ-IN-1
HY-120497-01	PKCζ-IN-1
HY-P3201	PKCζ/ι pseudosubstrate inhibitor
HY-162520	DJ-1-IN-1
HY-W176171-04	PU.1-IN-1
HY-W176171-02	PU.1-IN-1
HY-W176171-01	PU.1-IN-1
HY-U00003-07	ICAM-1-IN-1
HY-163731-06	EGR-1-IN-1
HY-163731-05	EGR-1-IN-1