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(R) -KT109

CAT: 0804-HY-126031-01Size: 500 µgDry Ice: NoHazardous: No
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CAT#:0804-HY-126031-01Size:500 µg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
(R) -KT109 is a highly potent inhibitor of diacylglycerol lipase β (DAGLβ) with an IC50 of 0.79 nM and effectively blocks DAGLα-mediated hydrolysis of 1-stearoyl-2-arachidonoyl-sn-glycerol. Additionally, it demonstrates inhibitory activity against α/β-hydrolase domain-containing protein 6 (ABHD6) with an IC50 of 2.51 nM, exhibiting greater potency for DAGLβ, DAGLα, and ABHD6 compared to its (S) isomer, (S) -KT109.
CAS Number
2055172-60-4
UNSPSC
12352005
Target
DAGL
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/r-kt109.html
Smiles
O=C(N1C=C(C2=CC=C(C3=CC=CC=C3)C=C2)N=N1)N4[C@H](CCCC4)CC5=CC=CC=C5
Molecular Formula
C27H26N4O
Molecular Weight
422.52
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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453073-01KT109
T38148-01(S) -KT109
T38031-01(R) -KT109
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