Nor-benzetimide

• Description :

  Nor-benzetimide is a major metabolite of Benzetimide. Benzetimide is a mAChR antagonist with anticholinergic activity[1][2].

• CAS Number :

  [19315-71-0]

• UNSPSC :

  12352005

• Target :

  MAChR

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Neuronal Signaling

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Neurological Disease

• Assay Protocol :

  https://www.medchemexpress.com/nor-benzetimide.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=C(C(C1CCNCC1)(C2=CC=CC=C2)CC3)NC3=O

• Molecular Formula :

  C16H20N2O2

• Molecular Weight :

  272.34

• References & Citations :

  [1] I van Wijngaarden. Differential anticholinergic activity, metabolism and excretion of the optical isomers of 14C-benzetimide hydrochloride. Life Sci. 1969 May 1;8 (9) :517-23.|[2]J A Gray, et al. Stereoselective binding in cardiac tissue of the enatiomers of benzetimide, and antimuscarinic drug. Br J Pharmacol. 1976 Apr;56 (4) :485-90.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported