HDAC/NAMPT-IN-1
CAT:
804-HY-162124
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

HDAC/NAMPT-IN-1
- CAS Number: 2898381-63-8
- UNSPSC Description: HDAC/NAMPT-IN-1 (compound 39h) is a dual inhibitor of HDAC and NAMPT with IC50 values of 0.72-37081 nM and 1618 nM[1].
- Target Antigen: HDAC; NAMPT
- Type: Reference compound
- Related Pathways: Cell Cycle/DNA Damage;Epigenetics;Metabolic Enzyme/Protease
- Applications: Cancer-programmed cell death
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/hdac-nampt-in-1.html
- Solubility: 10 mM in DMSO
- Smiles: CCCNNC(C1=CC=C(CNC(C2=CC3=CN=CC=C3N2)=O)C=C1)=O
- Molecular Weight: 351.40
- References & Citations: [1]Kairui Yue, et al. HDAC/NAMPT dual inhibitors overcome initial drug-resistance in p53-null leukemia cells. Eur J Med Chem. 2024.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported