Lenalidomide-acetylene-Br
CAT:
804-HY-156700
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For Laboratory Research Only. Not for Clinical or Personal Use.
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


Lenalidomide-acetylene-Br
UNSPSC Description:
Lenalidomide-acetylene-Br is a PROTAC Linker taht makes up HJM-561 (HY-156698). HJM-561 is a potent, selective, and orally active EGFR PROTAC to inhiibit Osimertinib (HY-15772)-resistant EGFR triple mutations.Target Antigen:
PROTAC LinkersType:
Reference compoundRelated Pathways:
PROTACApplications:
Cancer-programmed cell deathField of Research:
cancerAssay Protocol:
https://www.medchemexpress.com/lenalidomide-acetylene-br.htmlSolubility:
10 mM in DMSOSmiles:
O=C1NC(C(CC1)N2C(C3=C(C2)C(C#CCCBr)=CC=C3)=O)=OMolecular Weight:
375.22Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
2619512-84-2