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KSK67

CAT: 0804-HY-155615-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-155615-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
KSK67 is a high-affinity dual sigma-2 and histamine H3 receptor antagonist, with Kis of 3.2, 1531, 101 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK67 can be used for research of nociceptive and neuropathic pain[1].
CAS Number
2566715-93-1
UNSPSC
12352005
Target
Histamine Receptor; Sigma Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ksk67.html
Solubility
10 mM in DMSO
Smiles
O=C(C1CC1)C2=CC=C(OCCCN3CCN(C4=CC=NC=C4)CC3)C=C2
Molecular Formula
C22H27N3O2
Molecular Weight
365.47
References & Citations
[1]Szczepańska K, et al. Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain. J Med Chem. 2023 Jul 27;66 (14) :9658-9683.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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