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HPSE1-IN-1

CAT: 0804-HY-155410Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-155410Size:1 Each
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Description
HPSE1-IN-1 (compound 16) is a selective inhibitor of Heparanase-1 (HPSE1) with moderate inhibitory activity against exo-β-d-glucuronidase (GUSβ) and glucocerebrosidase (GBA) [1].
CAS Number
2876926-29-1
UNSPSC
12352005
Target
Endogenous Metabolite
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/hpse1-in-1.html
Solubility
10 mM in DMSO
Smiles
OC([C@H]1N2C([C@@H]([C@H]([C@@H]1OCCC3=CC=CC=C3)O)O)=NC(CCC4=CC(OC5=CC=CC=C5)=CC=C4)=C2)=O
Molecular Formula
C30H30N2O6
Molecular Weight
514.57
References & Citations
[1]Imai Y et al. Discovery of a novel tetrahydroimidazo [1, 2-a] pyridine-5-carboxylic acid derivative as a potent and selective heparanase-1 inhibitor utilizing an improved synthetic approach[J]. Bioorganic & Medicinal Chemistry Letters, 2023: 129543.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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