Casein kinase 1δ-IN-5
CAT:
804-HY-153904
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Casein kinase 1δ-IN-5
- CAS Number: 1579991-10-8
- UNSPSC Description: Casein kinase 1δ-IN-5 is a potent and selective protein kinase CK-1δ inhibitor with an IC50 of 47 nM. Casein kinase 1δ-IN-5 shows neuroprotective and anti-inflammatory properties both in vitro. Casein kinase 1δ-IN-5 has the potential for neurodegenerative diseases research.
- Target Antigen: Casein Kinase
- Type: Reference compound
- Related Pathways: Cell Cycle/DNA Damage;Stem Cell/Wnt
- Applications: Neuroscience-Neurodegeneration
- Field of Research: Neurological Disease
- Assay Protocol: https://www.medchemexpress.com/casein-kinase-1δ-in-5.html
- Solubility: 10 mM in DMSO
- Smiles: O=C(CC1=CC=CC=C1)NC2=NC3=C(S2)C=C(C(F)(F)F)C=C3
- Molecular Weight: 336.33
- References & Citations: [1]José A Morales-Garcia, et al. Biological and Pharmacological Characterization of Benzothiazole-Based CK-1δ Inhibitors in Models of Parkinson's Disease. ACS Omega
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported