PBRM1-BD2-IN-3

• UNSPSC Description:

  PBRM1-BD2-IN-3 (compound 12) is a potent PBRM1-BD2 inhibitor with an IC50 value of 1.1 μM. PBRM1-BD2 Inhibitor can be used to research anticancer[1].

• Target Antigen:

  Epigenetic Reader Domain

• Type:

  Reference compound

• Related Pathways:

  Epigenetics

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/pbrm1-bd2-in-3.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C1NC(C2=CC=CC=C2)NC3=C1C(Cl)=CC=C3

• Molecular Weight:

  258.70

• References & Citations:

  [1]Shishodia S, et al. Selective and Cell-Active PBRM1 Bromodomain Inhibitors Discovered through NMR Fragment Screening. J Med Chem. 2022 Oct 13.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2819989-58-5