Cavα2δ1&NET-IN-3
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804-HY-148866
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
Cavα2δ1&NET-IN-3
- CAS Number: 2143584-82-9
- UNSPSC Description: Cavα2δ1&NET-IN-3 (example 216) is an inhibitor of the subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has Kis of 100-500 nM for human α2δ-1 subunit of Cav2.2 calcium channel and NET, respectively[1].
- Target Antigen: Calcium Channel
- Type: Reference compound
- Related Pathways: Membrane Transporter/Ion Channel;Neuronal Signaling
- Applications: Metabolism-protein/nucleotide metabolism
- Field of Research: Endocrinology; Neurological Disease
- Assay Protocol: https://www.medchemexpress.com/cavα2δ1-net-in-3.html
- Solubility: 10 mM in DMSO
- Smiles: O=C1C2=CN=C(NCC)N=C2N(CCN1C3=CC(O[C@H](C4=CC=CS4)CCNC)=CC=C3)C
- Molecular Weight: 466.60
- References & Citations: [1]Félix CUEVAS-CORDOBÉS, et al. Tetrahydropyrimidodiazepine and tetrahydropyridodiazepine compounds for treating pain and pain related conditions. WO2017191304A1.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported