FAK-IN-8

• UNSPSC Description:

  FAK-IN-8 (compound 5h) is a FAK inhibitor (IC50=5.32 μM). FAK-IN-8 has good anti-proliferative activity and can be used in cancer research[1].

• Target Antigen:

  FAK

• Type:

  Reference compound

• Related Pathways:

  Protein Tyrosine Kinase/RTK

• Applications:

  Cancer-Kinase/protease

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/fak-in-8.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(NC1=NN=C(C2=CC=C(Cl)C=C2)S1)C3=CC(Cl)=CC=C3O

• Molecular Weight:

  366.22

• References & Citations:

  [1]Yang XH, et al. Synthesis, biological evaluation, and molecular docking studies of 1,3,4-thiadiazol-2-amide derivatives as novel anticancer agents. Bioorg Med Chem. 2012 May 1;20(9):2789-95.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  1374959-91-7