FAK-IN-7
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


FAK-IN-7
UNSPSC Description:
FAK-IN-7 (compound 5r) is a FAK inhibitor (IC50=11.72 μM). FAK-IN-7 has good anti-proliferative activity and can be used in cancer research[1].Target Antigen:
FAKType:
Reference compoundRelated Pathways:
Protein Tyrosine Kinase/RTKApplications:
Cancer-Kinase/proteaseField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/fak-in-7.htmlSolubility:
DMSO : 10 mg/mL (ultrasonic;warming;heat to 60°C)Smiles:
O=C(NC1=NN=C(C2=CC=C(C)C=C2)S1)C3=CC=CC=C3Molecular Weight:
295.36References & Citations:
[1]Yang XH, et al. Synthesis, biological evaluation, and molecular docking studies of 1,3,4-thiadiazol-2-amide derivatives as novel anticancer agents. Bioorg Med Chem. 2012 May 1;20(9):2789-95.Shipping Conditions:
Room TemperatureClinical Information:
No Development ReportedCAS Number:
19948-85-7
