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CXCR4 antagonist 9

CAT: 0804-HY-147979Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-147979Size:1 Each
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Description
CXCR4 antagonist 9 (Compound 2) is a CXCR4 antagonist with an IC50 of 15 nM. CXCR4 antagonist 9 inhibits CXCL12 induced cytosolic calcium increase with an IC50 of 1.3 nM[1].
CAS Number
2304750-83-0
UNSPSC
12352005
Target
CXCR
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation
Applications
COVID-19-immunoregulation
Field of Research
Cancer; Infection
Assay Protocol
https://www.medchemexpress.com/cxcr4-antagonist-9.html
Solubility
10 mM in DMSO
Smiles
CN1CCN(C2=CC(CN(C)C3=C(F)CCC4=C3N=CC=C4)=NC(C)=N2)CC1
Molecular Formula
C21H27FN6
Molecular Weight
382.48
References & Citations
[1]Lin Y, et al. Design, synthesis, and evaluation of novel CXCR4 antagonists based on an aminoquinoline template. Bioorg Chem. 2020 Jun;99:103824.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CXCR4

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