KCa1.1 channel activator-1

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804-HY-146173

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UNSPSC Description: KCa1.1 channel activator-1 (compound 1E), a Quercetin hybrid derivative, is a selective vascular KCa1.1 channel channel stimulator. KCa1.1 channel activator-1 also displays CaV1.2 channel blocking activity. KCa1.1 channel activator-1 exhibits weak myorelaxant activity[1].
Target Antigen: Calcium Channel; Potassium Channel
Type: Reference compound
Related Pathways: Membrane Transporter/Ion Channel;Neuronal Signaling
Applications: Neuroscience-Neuromodulation
Field of Research: Cardiovascular Disease
Assay Protocol: https://www.medchemexpress.com/kca1-1-channel-activator-1.html
Solubility: 10 mM in DMSO
Smiles: O=C(OC1=CC=C(C=C1O)C2=C(C(C3=C(O2)C=C(C=C3O)O)=O)O)/C=C/C4=CC=C5OCOC5=C4
Molecular Weight: 476.39
References & Citations: [1]Carullo G, et, al. Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular K Ca 1.1 channel stimulators. Bioorg Chem. 2020 Dec;105:104404.
Shipping Conditions: Room temperature
Clinical Information: No Development Reported

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