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A1AR antagonist 1

CAT: 0804-HY-144115Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-144115Size:1 Each
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Description
A1AR antagonist 1 (compound 18g) is a potent A1 adenosine receptor (AR) antagonist with Kis of 2.08, 6.91, and 31.2 nM for hA1, hA2A and hA2B, respectively[1].
CAS Number
2760128-99-0
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/a1ar-antagonist-1.html
Solubility
10 mM in DMSO
Smiles
NC1=NC(C2=CC(OC)=CC=C2)=C(C(C3=CC=CC=C3)=N1)C#N
Molecular Formula
C18H14N4O
Molecular Weight
302.33
References & Citations
[1]Val C, et al. Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1 Antagonists. J Med Chem. 2022;65 (3) :2091-2106.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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