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HA2AAR antagonist 1

CAT: 0804-HY-163701Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-163701Size:1 Each
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Description
HA2AAR antagonist 1 (compound 4a) is a highly selective hA2AAR antagonist with a Ki of 5 nM. hA2AAR antagonist 1 can be used in the study of immune-oncology[1].
CAS Number
2842150-81-4
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ha2aar-antagonist-1.html
Smiles
NC1=NC(C2=CC=CO2)=NC3=C1N=C(N3)C#CCCCC
Molecular Formula
C15H15N5O
Molecular Weight
281.31
References & Citations
[1]Kim G, et al. Structural Modification and Biological Evaluation of 2,8-Disubstituted Adenine and Its Nucleosides as A2A Adenosine Receptor Antagonists: Exploring the Roles of Ribose at Adenosine Receptors. J Med Chem. 2024 Jun 6.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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