WAY-207024 (dihydrochloride)

WAY-207024 (dihydrochloride)

• CAS Number: 872002-73-8
• UNSPSC Description: WAY-207024 (dihydrochloride) is a potent and orally active GnRH antagonist that reduces leuteinizing hormone (LH) levels in plasma[1].
• Target Antigen: GnRH Receptor
• Type: Reference compound
• Related Pathways: GPCR/G Protein
• Applications: Neuroscience-Neuromodulation
• Field of Research: Cardiovascular Disease
• Assay Protocol: https://www.medchemexpress.com/way-207024-dihydrochloride.html
• Solubility: 10 mM in DMSO
• Smiles: CC(C1=CC=C(C2=NC3=CC=CC(N4CCN(CC5=CC=C6N=CC=NC6=C5)CC4)=C3N2)C=C1)(C)C.[H]Cl.[H]Cl
• Molecular Weight: 549.54
• References & Citations: [1]Pelletier JC, et al. Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R). J Med Chem. 2009 Apr 9;52(7):2148-52.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported