CASK-IN-1

• UNSPSC Description:

  CASK-IN-1 is a highly potent and selective CASK inhibitor with a Kd value of 0.022 μM.

• Target Antigen:

  Others

• Type:

  Reference compound

• Related Pathways:

  Others

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/cask-in-1.html

• Purity:

  99.7

• Solubility:

  DMSO : 12.21 mg/mL (ultrasonic;warming)

• Smiles:

  O=C(C1=CN=C(N=C1NC2CCCC2)NCC3=CC(Br)=C(C=C3Br)C)NCCCN4CCOC4=O

• Molecular Weight:

  610.34

• References & Citations:

  [1]Russ N, et al. Design and Development of a Chemical Probe for Pseudokinase Ca2+/calmodulin-Dependent Ser/Thr Kinase. J Med Chem. 2021 Oct 14;64(19):14358-14376.

• Shipping Conditions:

  Blue Ice

• Storage Conditions:

  -20°C, 3 years (Powder)

• Clinical Information:

  No Development Reported

• CAS Number:

  2755241-73-5