SMYD2-IN-1

• UNSPSC Description:

  SMYD2-IN-1 is a SMYD2 inhibitor extracted from patent WO2016166186A1, compound example 1.1, has an IC50 of 4.45 nM[1].

• Target Antigen:

  Histone Methyltransferase

• Type:

  Reference compound

• Related Pathways:

  Epigenetics

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/smyd2-in-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  ClC1=CC(C2=NN(/C(NC3=CC=CC(OC(F)F)=C3)=N\C#N)CC2N(C([C@@H]4NCCC4)=O)CC)=CC=C1Cl

• Molecular Weight:

  564.41

• References & Citations:

  [1]Timo Stellfeld, et al. Novel aryl-cyanoguanidine compounds. WO2016166186A1.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2023788-96-5