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Sst2 Receptor agonist-1

CAT: 0804-HY-110161Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-110161Size:1 Each
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Description
Sst2 Receptor agonist-1 is a potent somatostatin receptor subtype 2 (sst2) agonist with a Ki value of 0.025 nM and a cAMP IC50 value of 4.8 nM. sst2 Receptor agonist-1 can inhibit rat growth hormone (GH) secretion and ocular neovascular lesion formation. Antiangiogenic effect[1].
CAS Number
1021912-42-4
UNSPSC
12352005
Target
Somatostatin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/sst2-receptor-agonist-1.html
Solubility
10 mM in DMSO
Smiles
ClC1=CC2=NC=C(C(OCCCN)=C2C=C1C3=CC=CC(O)=C3)C4=CC(C)=CC(C)=C4
Molecular Formula
C26H25ClN2O2
Molecular Weight
432.94
References & Citations
[1]Wolkenberg SE, et al. Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2. J Med Chem. 2011 Apr 14;54 (7) :2351-8.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
SSTR2

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