PDK1-IN-3

• UNSPSC Description:

  PDK1-IN-3 (Compound C) is a PDK1 inhibitor, with an IC50 of 34 nM[1].

• Target Antigen:

  PDK-1

• Type:

  Reference compound

• Related Pathways:

  PI3K/Akt/mTOR

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/pdk1-in-3.html

• Smiles:

  N#CCC(C=C1)=CC=C1N2C=NC3=C2C4=CC(C#CC5=CC=CN=C5)=CC=C4N=C3

• Molecular Weight:

  385.42

• References & Citations:

  [1]Murphy ST, et al. Discovery of novel, potent, and selective inhibitors of 3-phosphoinositide-dependent kinase (PDK1). J Med Chem. 2011 Dec 22;54(24):8490-500.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  853909-77-0