R-84760

• UNSPSC Description:

  R-84760 is a selective κ-opioid receptor agonist. R-84760 has antinociceptive effect[1][2].

• Target Antigen:

  Opioid Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Neuronal Signaling

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/r-84760.html

• Smiles:

  O=C([C@H]1CCC2=C1C=C(Cl)C(Cl)=C2)N3[C@H](CN4CCCC4)CSCC3.Cl

• Molecular Weight:

  435.84

• References & Citations:

  [1]Fujibayashi K, et al. Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist.[J].European Journal of Pharmacology, 1994, 261(1-2):133-140.|[2]Fujibayashi K, et al. Profiles of the antinociceptive effect of R-84760, a selective kappa-opioid receptor agonist, in the formalin test in mice. Jpn J Pharmacol. 1995 May;68(1):57-63.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  Phase 2

• CAS Number:

  157824-23-2