Eplivanserin (mixture)

• Description:

  Eplivanserin mixture (SR-46349 mixture) is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1[1].

• Product Name Alternative:

  SR-46349 (mixture)

• UNSPSC:

  12352005

• Target:

  5-HT Receptor; Serotonin Transporter

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/eplivanserin-mixture.html

• Purity:

  99.68

• Solubility:

  DMSO : 125 mg/mL (ultrasonic)

• Smiles:

  OC1=CC=C (/C=C/C (C2=CC=CC=C2F) =N/OCCN (C) C) C=C1

• Molecular Formula:

  C19H21FN2O2

• Molecular Weight:

  328.38

• References & Citations:

  [1]BERMAN, Robert, Mark, et al. COMPOSITIONS CONTAINING A SEROTONIN SELECTIVE REUPTAKE INHIBITOR AND A 5-HT2A RECEPTOR ANTAGONIST. WO 2005/002578 A1.

• Shipping Conditions:

  Room Temperature

• Storage Conditions:

  -20°C, 3 years; 4°C, 2 years (Powder)

• Scientific Category:

  Reference compound1

• Clinical Information:

  Phase 3

• Isoform:

  5-HT2 Receptor; α-1 microglobulin

• CAS Number:

  130581-13-4