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Pitolisant-d5 (hydrochloride)

CAT: 0804-HY-12199BSSize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-12199BSSize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Pitolisant-d5 hydrochloride (Ciproxidine-d5 hydrochloride) is the deuterium labeled Pitolisant hydrochloride. Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
CAS Number
2740634-42-6
Product Name Alternative
Ciproxidine-d5 (hydrochloride) ; BF 2649-d5 (hydrochloride)
UNSPSC
12352005
Target
Histamine Receptor; Isotope-Labeled Compounds
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling; Others
Field of Research
Endocrinology; Neurological Disease
Smiles
ClC(C=C1)=CC=C1C([2H])C([2H])([2H])C([2H])([2H])OCCCN2CCCCC2.Cl
Molecular Formula
C17H22D5Cl2NO
Molecular Weight
337.34
References & Citations
[1]Ligneau X, et al. BF2.649 [1-{3-[3- (4-Chlorophenyl) propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology. J Pharmacol Exp Ther. 2007 Jan;320 (1) :365-75.|[2]Dudek M, et al. H3 histamine receptor antagonist pitolisant reverses some subchronic disturbances induced by LY170053 in mice. Metab Brain Dis. 2016 Oct;31 (5) :1023-9.|[3]Uguen M, et al. Preclinical evaluation of the abuse potential of Pitolisant, a histamine H? receptor inverse agonist/antagonist compared with CRL 40476. Br J Pharmacol. 2013 Jun;169 (3) :632-44.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported

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CS-O-41499Pitolisant D5 Hydrochloride
A3727-5.1Pitolisant hydrochloride
A15213-5Pitolisant hydrochloride 5mg
TRC-H107260-50MGHydroxy Pitolisant Hydrochloride
A15213-200Pitolisant hydrochloride 200mg
A15213-50Pitolisant hydrochloride 50mg
A15213-10Pitolisant hydrochloride 10mg
A15213-100Pitolisant hydrochloride 100mg
A15213-25Pitolisant hydrochloride 25mg
A15213-500Pitolisant hydrochloride 500mg

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