Products for Research Use Only
RegisterLogin

R-138727

CAT: 0804-HY-123669Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-123669Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
R-138727, the thiol-containing active metabolite of Prasugrel, is an irreversible platelet P2Y12 receptor inhibitor. R-138727 inhibits ADP-induced platelet aggregation[1].
CAS Number
204204-73-9
UNSPSC
12352005
Target
Drug Metabolite; P2Y Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/r-138727.html
Solubility
10 mM in DMSO
Smiles
O=C(/C=C1CN(CCC/1S)C(C(C2CC2)=O)C3=CC=CC=C3F)O
Molecular Formula
C18H20FNO3S
Molecular Weight
349.42
References & Citations
[1]Hasegawa M, et al. Stereoselective inhibition of human platelet aggregation by R-138727, the active metabolite of CS-747 (prasugrel, LY640315), a novel P2Y12 receptor inhibitor. Thromb Haemost. 2005 Sep;94 (3) :593-8.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-123669AS-01(R) -trans-138727-d4
HY-W998245(R, R, R) -AHPC (hydrochloride)
HY-W018061C-01(R, R) -Traxoprodil
HY-103451(R, R) -THC
HY-128888-01(R, R) -GSK321
HY-113834(R, R) -Ethambutol
HY-59125-01(R, R) - (+) -Hydrobenzoin
HY-100443B-01(R, R) -PX20606
HY-B0761(R, R) -Glycopyrrolate
HY-100741C-01(R, R) -S63845

Alternative Products

CatalogName
MBS5772093R-138727
BA5682-1trans-R-138727
AR-P29568-01Prasugrel Metabolite R-138727
CS-O-64435Prasugrel Metabolite R-138727-d4
AR-P02508-01Prasugrel-d4 Metabolite R-138727
CS-O-56605Trans R-138727 (Prasugrel Metabolite)
AR-P32359-01Prasugrel Metabolite R-138727 HCl (Mixture of Diastereomers)
TRC-R070195-5MGtrans R-138727, (Prasugrel Metabolite) - >90%(Mixture of Diastereomers)
467773-01Trans R-138727, (Prasugrel Metabolite) - >90% (Mixture of Diastereomers)
467772Trans R-138727-d4, (Prasugrel-d4 Metabolite) (Mixture of Diastereomers)

Popular Products