Bilaid C

• Description:

  Bilaid C, a tetrapeptide, can be isolated from the Australian estuarine isolate of Penicillium sp. MST-MF667. Bilaid C is also a potent and selective μ-Opioid Receptor (MOPr) agonist (Ki=210 nM, hMOPr) [1].

• UNSPSC:

  12352209

• Target:

  Opioid Receptor

• Type:

  Peptides

• Related Pathways:

  GPCR/G Protein; Neuronal Signaling

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/bilaid-c.html

• Solubility:

  10 mM in DMSO

• Smiles:

  OC(C=C1)=CC=C1C[C@H](N)C(N[C@H](C(C)C)C(N[C@@H](C(C)C)C(N[C@@H](C(O)=O)CC2=CC=CC=C2)=O)=O)=O

• Molecular Formula:

  C28H38N4O6

• Molecular Weight:

  526.62

• References & Citations:

  [1]Dekan Z, et al. A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor. Proc Natl Acad Sci U S A. 2019 Oct 29;116 (44) :22353-22358.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Peptides

• Clinical Information:

  No Development Reported

• Isoform:

  μ Opioid Receptor/MOR

• CAS Number:

  [2393866-13-0]