Protease-Activated Receptor-2, amide

Protease-Activated Receptor-2, amide

• CAS Number: 190383-13-2
• UNSPSC Description: Protease-Activated Receptor-2, amide (SLIGKV-NH2) is a highly potent protease-activated receptor-2 (PAR2) activating peptide.
• Target Antigen: Protease Activated Receptor (PAR)
• Type: Peptides
• Related Pathways: GPCR/G Protein
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/Protease-Activated_Receptor-2,_amide.html
• Purity: 98.73
• Solubility: H2O : 33.33 mg/mL (ultrasonic)
• Smiles: CC(C)[C@@H](C(N)=O)NC([C@H](CCCCN)NC(CNC([C@H]([C@@H](C)CC)NC([C@H](CC(C)C)NC([C@H](CO)N)=O)=O)=O)=O)=O
• Molecular Weight: 614.78
• References & Citations: [1]Kanke T, et al. Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [3H]2-furoyl-LIGRL-NH2, to human PAR2. Br J Pharmacol. 2005 May;145(2):255-63.|[2]Ramelli G, et al. Protease-activated receptor 2 signalling promotes dendritic cell antigen transport and T-cellactivation in vivo. Immunology. 2010 Jan;129(1):20-7.
• Shipping Conditions: Blue Ice
• Storage Conditions: -80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
• Clinical Information: No Development Reported