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(Rac) -Acolbifene

CAT: 0804-HY-16023B-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-16023B-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
(Rac) -Acolbifene (EM-343; (Rac) -EM-652) is the racemic form of EM652 (estrogen receptor antagonist), has anti-estrogenic and estrogenic activities. (Rac) -Acolbifene (EM-343; (Rac) -EM-652) contains a piperidine ring, shows good pharmacological profile, relative binding affinity (RBA) =380[1].
CAS Number
151533-34-5
Product Name Alternative
EM-343; (Rac) -EM-652
UNSPSC
12352005
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/rac-acolbifene.html
Concentration
10mM
Purity
98.18
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
OC1=CC=C2C(C)=C(C3=CC=C(O)C=C3)C(C4=CC=C(OCCN5CCCCC5)C=C4)OC2=C1
Molecular Formula
C29H31NO4
Molecular Weight
457.56
References & Citations
[1]Gauthier S1, et al.Synthesis and structure-activity relationships of analogs of EM-652 (acolbifene), a pure selective estrogen receptor modulator. Study of nitrogen substitution.J Enzyme Inhib Med Chem. 2005 Apr;20 (2) :165-77.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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