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Endomorphin 2 (TFA)

CAT: 0804-HY-P0186A-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-P0186A-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].
CAS Number
1276124-00-5
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/endomorphin-2-tfa.html
Purity
99.04
Solubility
DMSO : < 1 mg/mL|H2O : 125 mg/mL (ultrasonic)
Smiles
O=C(N)[C@H](CC1=CC=CC=C1)NC([C@H](CC2=CC=CC=C2)NC([C@H]3N(C([C@H](CC4=CC=C(C=C4)O)N)=O)CCC3)=O)=O.OC(C(F)(F)F)=O
Molecular Formula
C34H38F3N5O7
Molecular Weight
685.69
References & Citations
[1]Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286 (2) :1007-13.
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
μ Opioid Receptor/MOR