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Brompheniramine (Standard)

CAT: 0804-HY-B0480ARSize: 1 EachDry Ice: NoHazardous: No
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Description
Brompheniramine (Standard) is the analytical standard of Brompheniramine. This product is intended for research and analytical applications. Brompheniramine ((±) -Brompheniramine) is a potent and orally active antihistamine of the alkylamine class. Brompheniramine is a selective histamine H1 receptor antagonist with a Kd of 6.06 nM. Brompheniramine can block the hERG channels, calcium channels, and sodium channels with IC50s of 0.90 μM, 16.12 μM and 21.26 μM, respectively. Brompheniramine has anticholinergic, antidepressant and anesthetic properties and can be used for allergic rhinitis research[1][2][3][4].
CAS Number
86-22-6
Product Name Alternative
(±) -Brompheniramine (Standard)
UNSPSC
12352005
Target
Calcium Channel; Histamine Receptor; mAChR; Potassium Channel; Reference Standards; Sodium Channel
Type
Reference Standards
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Membrane Transporter/Ion Channel; Neuronal Signaling; Others
Field of Research
Endocrinology; Inflammation/Immunology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/brompheniramine-standard.html
Smiles
CN(C)CCC(C1=CC=C(Br)C=C1)C2=CC=CC=N2
Molecular Formula
C16H19BrN2
Molecular Weight
319.24
References & Citations
[1]Chong-Chi Chiu, et al. Subcutaneous brompheniramine for cutaneous analgesia in rats. Eur J Pharmacol. 2019 Oct 5;860:172544.|[2]B Cusack, et al. Binding of antidepressants to human brain receptors: focus on newer generation compounds. Psychopharmacology (Berl) . 1994 May;114 (4) :559-65.|[3]Shin WH, Kim KS, Kim EJ. Electrophysiological effects of brompheniramine on cardiac ion channels and action potential. Pharmacol Res. 2006 Dec;54 (6) :414-20.|[4]Yasuda SU, Yasuda RP. Affinities of brompheniramine, chlorpheniramine, and terfenadine at the five human muscarinic cholinergic receptor subtypes. Pharmacotherapy. 1999 Apr;19 (4) :447-51.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards

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