DDR2-IN-1

DDR2-IN-1

• CAS Number: 1573053-23-2
• UNSPSC Description: DDR2-IN-1 is potent DDR2 inhibitor with an IC50 of 26 nM. DDR2-IN-1, compound 129, can be used for osteoarthritis research[1].
• Target Antigen: Discoidin Domain Receptor
• Type: Reference compound
• Related Pathways: Protein Tyrosine Kinase/RTK
• Applications: Metabolism-protein/nucleotide metabolism
• Field of Research: Metabolic Disease
• Assay Protocol: https://www.medchemexpress.com/ddr2-in-1.html
• Purity: 99.88
• Solubility: DMSO : 250 mg/mL (ultrasonic)
• Smiles: O=C(C1=NC=CC(OC2=CC=C(CNC(NC3=CC(C)=C(Cl)C=C3OCCN(C)C)=O)C=C2C)=C1)NC
• Molecular Weight: 526.03
• References & Citations: [1]Margarita Wucherer-Plietker, et al. Inhibiteurs de ddr2 pour le traitement de l'arthrose. Patent WO2014032755A2.
• Shipping Conditions: Room Temperature
• Storage Conditions: -20°C, 3 years; 4°C, 2 years (Powder)
• Clinical Information: No Development Reported